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Journal of Medicinal Chemistry

Syndicate content Journal of Medicinal Chemistry: Latest Articles (ACS Publications)
Table of Contents for Journal of Medicinal Chemistry. List of articles from both the latest and ahead of print issues.
Updated: 1 day 18 hours ago

Single-Step High-Yield Radiosynthesis and Evaluation of a Sensitive 18F-Labeled Ligand for Imaging Brain Peripheral Benzodiazepine Receptors with PET

Fri, 01/02/2009 - 9:22am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Revision of Purity Criteria for Tested Compounds

Fri, 01/02/2009 - 12:00am
Journal of Medicinal Chemistry, Volume 52, Issue 1, Page 1, January 8, 2009.
Categories: ACS Publications

Synthesis of Novel 4,6-Di(substituted)amino-1,2-dihydro-1,3,5-triazine Derivatives as Topical Antiseptic Agents

Wed, 12/31/2008 - 12:12pm
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Design, Synthesis, and Evaluation in Vitro of Quinoline-8-carboxamides, a New Class of Poly(adenosine-diphosphate-ribose)polymerase-1 (PARP-1) Inhibitor

Wed, 12/31/2008 - 11:29am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Structure−Activity Relationship and Studies on the Molecular Mechanism of Leishmanicidal N,C-Coupled Arylisoquinolinium Salts

Wed, 12/31/2008 - 11:26am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Design, Synthesis, and Biological Evaluation of Fluorinated Analogues of Salicylihalamide

Wed, 12/31/2008 - 9:47am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

First Cdc7 Kinase Inhibitors: Pyrrolopyridinones as Potent and Orally Active Antitumor Agents. 2. Lead Discovery†

Tue, 12/30/2008 - 10:52am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Fragment-Based Discovery of the Pyrazol-4-yl Urea (AT9283), a Multitargeted Kinase Inhibitor with Potent Aurora Kinase Activity†

Tue, 12/30/2008 - 10:51am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

6-Methoxy-N-alkyl Isatin Acylhydrazone Derivatives as a Novel Series of Potent Selective Cannabinoid Receptor 2 Inverse Agonists: Design, Synthesis, and Binding Mode Prediction

Tue, 12/30/2008 - 8:44am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Synthesis, Oxidant Properties, and Antitumoral Effects of a Heteroleptic Palladium(II) Complex of Curcumin on Human Prostate Cancer Cells

Mon, 12/29/2008 - 4:52pm
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Synthesis and Biological Studies of Different Duocarmycin Based Glycosidic Prodrugs for Their Use in the Antibody-Directed Enzyme Prodrug Therapy

Mon, 12/29/2008 - 4:49pm
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Combining 4-Aminoquinoline- and Clotrimazole-Based Pharmacophores toward Innovative and Potent Hybrid Antimalarials

Mon, 12/29/2008 - 3:26pm
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Edaravone Derivatives Containing NO-Donor Functions

Mon, 12/29/2008 - 3:24pm
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Design, Structure−Activity Relationships and in Vivo Characterization of 4-Amino-3-benzimidazol-2-ylhydroquinolin-2-ones: A Novel Class of Receptor Tyrosine Kinase Inhibitors

Mon, 12/29/2008 - 11:22am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Dual Integrin and Gastrin-Releasing Peptide Receptor Targeted Tumor Imaging Using 18F-labeled PEGylated RGD-Bombesin Heterodimer 18F-FB-PEG3-Glu-RGD-BBN

Mon, 12/29/2008 - 11:11am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Discovery of Novel CB2 Receptor Ligands by a Pharmacophore-Based Virtual Screening Workflow

Mon, 12/29/2008 - 11:07am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Induced Association of μ Opioid (MOP) and Type 2 Cholecystokinin (CCK2) Receptors by Novel Bivalent Ligands

Mon, 12/29/2008 - 11:04am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications

Synthesis and Biological Activity of Human Neuropeptide S Analogues Modified in Position 5: Identification of Potent and Pure Neuropeptide S Receptor Antagonists

Mon, 12/29/2008 - 11:03am
Journal of Medicinal Chemistry, Volume 0, Issue 0, Articles ASAP (As Soon As Publishable).
Categories: ACS Publications